SCHEMBL8035622

SCHEMBL8035622

CCCNC(=O)N(C)C(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
COMT P21964 4/20 0.37
POLB P06746 2/20 0.32
ERN1 O75460 1/20 0.32
ALDH1A1 P00352 4/20 0.31
KMT2A Q03164 4/20 0.31
MEN1 O00255 3/20 0.31
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPT P10636 2/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025508 0.87 ALDH1A1 (0.37) COMTPOLBALDH1A1KMT2ALMNA
SCHEMBL8041249 0.81 TAS1R3 (0.35) COMTALDH1A1
SCHEMBL8039069 0.74 COMT (0.40) COMTALDH1A1KMT2AMEN1LMNA
SCHEMBL8041625 0.74 EGFR (0.35) POLBERN1ALDH1A1KMT2AMEN1
SCHEMBL8041245 0.74 MAPT (0.39) COMTPOLBALDH1A1KMT2AMEN1
SCHEMBL8037862 0.74 CYP3A4 (0.38) COMTALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL8035693 0.73 HSP90AA1 (0.35) COMTPOLBKMT2AMEN1
SCHEMBL8041445 0.73 EPHX2 (0.41)
SCHEMBL8035781 0.73 EPHX2 (0.41)
SCHEMBL8041408 0.70 SMN1; SMN2 (0.32) COMTPOLBALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed