SCHEMBL8038899

SCHEMBL8038899

O=C(NCc1ccccc1)NC(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.52
TP53 P04637 1/20 0.44
MITF O75030 1/20 0.43
KMT2A Q03164 5/20 0.40
MEN1 O00255 4/20 0.40
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041445 0.78 EPHX2 (0.41)
SCHEMBL8041408 0.78 SMN1; SMN2 (0.32) KMT2AMEN1MAPTALDH1A1POLB
SCHEMBL8025495 0.77 KMT2A (0.48) KMT2AMEN1MAPTALDH1A1POLB
SCHEMBL8037861 0.76 PPIA (0.41) PPIAMAPTALDH1A1POLBL3MBTL1
SCHEMBL8040243 0.74 PPIA (0.47) PPIAKMT2AMEN1MAPTALDH1A1
SCHEMBL8025492 0.74 PPIA (0.49) PPIAKMT2AMEN1MAPTALDH1A1
SCHEMBL8037250 0.72 TAS1R3 (0.45) PPIAMAPTALDH1A1HPGDKDM4E
SCHEMBL8035160 0.71 KMT2A (0.39) KMT2AMEN1MAPTALDH1A1L3MBTL1
SCHEMBL8037862 0.71 CYP3A4 (0.38) MAPTALDH1A1CYP3A4HTTNPSR1
SCHEMBL8035106 0.70 COMT (0.36) KMT2AMEN1MAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed