SCHEMBL8040243

SCHEMBL8040243

O=C(NC(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-])NC1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.47
MAPT P10636 3/20 0.41
GAA P10253 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
EPHX1 P07099 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RAB9A P51151 3/20 0.38
EPHX2 P34913 2/20 0.38
NPC1 O15118 1/20 0.38
THRB P10828 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025492 0.99 PPIA (0.49) PPIAMAPTGAAALDH1A1HPGD
SCHEMBL8037861 0.96 PPIA (0.41) PPIAMAPTGAAALDH1A1HPGD
SCHEMBL8037250 0.91 TAS1R3 (0.45) PPIAMAPTGAAALDH1A1HPGD
SCHEMBL8038220 0.86 PPIA (0.42) PPIAMAPTGAAALDH1A1KDM4E
SCHEMBL8025559 0.82 MAPT (0.37) PPIAMAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL8035603 0.80 RAB9A (0.40) MAPTALDH1A1SMN1; SMN2RAB9ANPC1
SCHEMBL8035160 0.79 KMT2A (0.39) MAPTGAAALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL8035162 0.77 ALDH1A1 (0.41) PPIAALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL8041249 0.75 TAS1R3 (0.35) ALDH1A1
SCHEMBL8025495 0.74 KMT2A (0.48) MAPTALDH1A1SMN1; SMN2RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed