SCHEMBL8039005

SCHEMBL8039005

COc1cc(Cl)c(C(=O)N(C)C(=O)NCc2ccc(N)cc2)cc1O

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.41
ALDH1A1 P00352 1/20 0.41
MMP9 P14780 1/20 0.40
HSP90AA1 P07900 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037001 0.83 ALDH1A1 (0.46) ALDH1A1
SCHEMBL8039016 0.82 HTT (0.42) TRPV1ALDH1A1HSP90AA1
SCHEMBL8035589 0.80 TRPV1 (0.41) TRPV1ALDH1A1HSP90AA1
SCHEMBL8041247 0.78 HSP90AA1 (0.39) TRPV1ALDH1A1HSP90AA1
SCHEMBL8035119 0.78 KDM4E (0.40) ALDH1A1HSP90AA1
SCHEMBL8035729 0.77 PTPN1 (0.37) ALDH1A1
SCHEMBL8035099 0.77 TRPV1 (0.47) TRPV1
SCHEMBL8039002 0.75 MAPT (0.39) ALDH1A1HSP90AA1
SCHEMBL8025491 0.74 KDM4E (0.42) ALDH1A1
SCHEMBL8032092 0.73 ALDH1A1 (0.44) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed