SCHEMBL8032092

SCHEMBL8032092

COc1cc(Cl)c(C(=O)N(C)C(=O)NC2CC2)cc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HTT P42858 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
HTR4 Q13639 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 2/20 0.39
KMT2A Q03164 2/20 0.39
GFER P55789 1/20 0.38
MAPT P10636 4/20 0.37
KDM4E B2RXH2 3/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
NOD2 Q9HC29 1/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031695 0.85 ALDH1A1 (0.43) ALDH1A1HTTTAS1R3TAS1R1TAS1R2
SCHEMBL8035119 0.83 KDM4E (0.40) ALDH1A1SMN1; SMN2KMT2AMAPTKDM4E
SCHEMBL8034162 0.82 LRRK2 (0.38) ALDH1A1HTTTAS1R3TAS1R1TAS1R2
SCHEMBL8039002 0.80 MAPT (0.39) ALDH1A1HTTTAS1R3TAS1R1TSHR
SCHEMBL8039016 0.80 HTT (0.42) ALDH1A1HTTSMN1; SMN2GFERKDM4E
SCHEMBL8025474 0.79 TSHR (0.39) TSHRKMT2AMAPTKDM4EHPGD
SCHEMBL8037071 0.79 MEN1 (0.47) ALDH1A1KMT2AMEN1NPC1LMNA
SCHEMBL8035589 0.78 TRPV1 (0.41) ALDH1A1HTTHTR4TSHRPOLB
SCHEMBL8040249 0.78 PYGL (0.47) ALDH1A1HTTTAS1R3TAS1R1TAS1R2
SCHEMBL8034159 0.78 ALDH1A1 (0.44) ALDH1A1HTTTSHRSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed