SCHEMBL8039002

SCHEMBL8039002

COc1cc(Cl)c(C(=O)N(C)C(=O)NC(C)C)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
CXCL12 P48061 3/20 0.37
LMNA P02545 2/20 0.36
HPGD P15428 2/20 0.36
HSP90AA1 P07900 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
NOD2 Q9HC29 1/20 0.36
GAA P10253 1/20 0.36
CYP3A4 P08684 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035119 0.85 KDM4E (0.40) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL8039016 0.82 HTT (0.42) ALDH1A1HTTSMN1; SMN2CXCL12LMNA
SCHEMBL8025473 0.81 HSP90AA1 (0.37) MAPTMEN1KMT2AALDH1A1HTT
SCHEMBL8032092 0.80 ALDH1A1 (0.44) MAPTMEN1KMT2AALDH1A1HTT
SCHEMBL8035589 0.80 TRPV1 (0.41) KMT2AALDH1A1HTTCXCL12LMNA
SCHEMBL8025491 0.79 KDM4E (0.42) MAPTMEN1KMT2AALDH1A1HTT
SCHEMBL8041247 0.78 HSP90AA1 (0.39) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL8038345 0.78 HPGD (0.52) MEN1KMT2AALDH1A1HTTSMN1; SMN2
SCHEMBL8039013 0.78 ALDH1A1 (0.41) MEN1KMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL8035099 0.77 TRPV1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed