SCHEMBL8039231

SCHEMBL8039231

COc1cc(Cl)c(C(=O)N(C)C(=O)NCC(F)(F)F)cc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.43
CTSL P07711 2/20 0.43
APP P05067 3/20 0.42
RAF1 P04049 1/20 0.42
MAP2K1 Q02750 1/20 0.42
EGFR P00533 1/20 0.42
SRD5A1 P18405 1/20 0.41
SRD5A2 P31213 1/20 0.41
SMPD1 P17405 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HPGD P15428 3/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035938 0.88 SRD5A1 (0.47) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8032086 0.86 NPC1 (0.47) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8034163 0.86 CTSV (0.47) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8038348 0.84 MTNR1A (0.47) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8038345 0.83 HPGD (0.52) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8037001 0.83 ALDH1A1 (0.46) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8032065 0.83 MTNR1A (0.46) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8037235 0.82 SMPD1 (0.45) CTSVCTSLEGFRSRD5A1SRD5A2
SCHEMBL8037071 0.82 MEN1 (0.47) CTSVCTSLAPPRAF1MAP2K1
SCHEMBL8032570 0.81 KDM4E (0.45) CTSVCTSLAPPRAF1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed