SCHEMBL8039263

SCHEMBL8039263

CCCNC(=O)c1cc(OCc2ccccc2)c(OC)cc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
SMPD1 P17405 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
HPGD P15428 3/20 0.46
ALDH1A1 P00352 2/20 0.46
BRD4 O60885 1/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
ROCK2 O75116 1/20 0.44
SGMS2 Q8NHU3 1/20 0.44
APP P05067 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025540 0.92 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8039245 0.92 MRGPRX4 (0.49) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8023140 0.90 MTNR1B (0.49) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8034962 0.89 HPGD (0.58) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8037062 0.87 SMPD1 (0.51) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8034976 0.86 NPC1 (0.45) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8039086 0.86 MTNR1A (0.47) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8037331 0.85 MTNR1A (0.46) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8041284 0.85 MTNR1A (0.46) SMN1; SMN2NPC1RAB9ASMPD1HDAC1
SCHEMBL8035471 0.84 CTSV (0.54) SMN1; SMN2NPC1RAB9ASMPD1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed