SCHEMBL8039635

SCHEMBL8039635

COc1ccc2ccc3c(c2c1)CCN=C3C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
CYP3A4 P08684 5/20 0.56
MEN1 O00255 3/20 0.56
CYP2D6 P10635 3/20 0.56
CASP1 P29466 3/20 0.56
KMT2A Q03164 3/20 0.56
HTR7 P34969 3/20 0.56
HTR2A P28223 2/20 0.56
HTR2C P28335 2/20 0.56
RECQL P46063 2/20 0.56
HTR6 P50406 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
CYP1A2 P05177 2/20 0.56
ALOX15 P16050 1/20 0.56
HSD17B10 Q99714 4/20 0.52
ALDH1A1 P00352 3/20 0.52
GLA P06280 2/20 0.52
HPGD P15428 2/20 0.52
TSHR P16473 2/20 0.52
CASP7 P55210 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875288 0.76 ALDH1A1 (0.60) KDM4ECYP3A4MEN1CYP2D6CASP1
Hydrochloric Acid SCHEMBL10662272 0.75 ALDH1A1 (0.58) KDM4ECYP3A4MEN1CYP2D6CASP1
SCHEMBL29664763 0.73 MAOA (0.60) KDM4ECYP3A4MEN1CYP2D6CASP1
SCHEMBL1010356 0.73 MAOA (0.60) KDM4ECYP3A4MEN1CYP2D6CASP1
SCHEMBL3877767 0.71 KDM4E (1.00) KDM4ECYP3A4MEN1CYP2D6CASP1
SCHEMBL1007423 0.69 KDM4E (0.54) KDM4EHTR2CALDH1A1HPGDGAA
SCHEMBL11831581 0.69 CA1 (0.46) KDM4ECYP3A4MEN1CYP2D6CASP1
SCHEMBL19382614 0.69 CYP1A2 (0.61) KDM4EMEN1KMT2AHTR2ACYP1A2
Harmaline SCHEMBL29626541 0.69 KDM4E (1.00) KDM4ECYP3A4MEN1CYP2D6CASP1
Harmaline SCHEMBL199260 0.69 KDM4E (1.00) KDM4ECYP3A4MEN1CYP2D6CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048868-A CIRCADIAN RHYTHM DISORDERS; SLEEP DISORDERS; ANTIDEPRESSANTS CEMAF (FR) 2000-04-11 US disclosed