SCHEMBL8039833

SCHEMBL8039833

CC(N)C1Cc2cc(Br)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 4/20 0.39
ADRA2A P08913 3/20 0.39
ADRA2B P18089 3/20 0.39
ADRA2C P18825 3/20 0.39
PBRM1 Q86U86 1/20 0.39
GLS O94925 2/20 0.34
KDM1A O60341 2/20 0.34
MAPT P10636 3/20 0.33
AHR P35869 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
NFKB1 P19838 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
HIF1A Q16665 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12303262 0.87 PNMT (0.44) PNMTADRA2AADRA2BADRA2CPBRM1
SCHEMBL8042044 0.82 AKT1 (0.35) MAPTTDP1MEN1ALDH1A1KMT2A
SCHEMBL10367511 0.78 ADRA2A (0.35) PNMTADRA2AADRA2BADRA2CPBRM1
SCHEMBL8899294 0.77 PNMT (0.37) PNMTKDM1A
SCHEMBL8042060 0.76 CYP19A1 (0.43) HTR2A
SCHEMBL8036024 0.76 CYP19A1 (0.43) HTR2A
SCHEMBL8038143 0.76 CYP19A1 (0.43) HTR2A
SCHEMBL8038148 0.76 CYP19A1 (0.43) HTR2A
SCHEMBL8042053 0.76 CYP19A1 (0.43) HTR2A
SCHEMBL8035992 0.75 PNMT (0.45) PNMTADRA2AADRA2BADRA2CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000076990-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-12-21 WO disclosed