SCHEMBL8040180

SCHEMBL8040180

COc1cc(C(F)(F)F)c(C(=O)NC(=O)Nc2ccccc2)cc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.58
ADRB2 P07550 1/20 0.52
GPR183 P32249 1/20 0.52
APLNR P35414 1/20 0.52
S1PR5 Q9H228 1/20 0.52
NPSR1 Q6W5P4 2/20 0.51
MAPT P10636 3/20 0.49
TP53 P04637 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ATM Q13315 1/20 0.49
THRB P10828 1/20 0.48
KDM4E B2RXH2 4/20 0.48
MAPK1 P28482 1/20 0.47
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALDH1A1 P00352 1/20 0.45
RCE1 Q9Y256 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033845 0.84 ATM (0.56) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8035613 0.83 S1PR1 (0.54) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8037361 0.82 S1PR1 (0.48) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8037447 0.81 S1PR1 (0.41) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8037438 0.80 S1PR1 (0.45) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8037366 0.80 S1PR1 (0.41) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8036048 0.80 KDM1A (0.43) S1PR1NPSR1MAPTTP53RAB9A
SCHEMBL8035722 0.78 RAB9A (0.52) S1PR1MAPTTP53NPC1RAB9A
SCHEMBL8037415 0.78 S1PR1 (0.41) S1PR1ADRB2GPR183APLNRS1PR5
SCHEMBL8040252 0.78 ALDH1A1 (0.41) S1PR1MAPTKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed