SCHEMBL8037366

SCHEMBL8037366

COc1cc(C(F)(F)F)c(C(=O)NC(=O)N(C)c2ccccc2)cc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
POLQ O75417 4/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ADRB2 P07550 1/20 0.38
GPR183 P32249 1/20 0.38
APLNR P35414 1/20 0.38
S1PR5 Q9H228 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.37
ALDH1A1 P00352 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028301 0.85 APP (0.39) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8035717 0.84 ALDH1A1 (0.45) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8041684 0.83 SMPD1 (0.44) KDM4EHPGDRXFP1MEN1KMT2A
SCHEMBL8022424 0.81 LMNA (0.42) KDM4ELMNACYP3A4MAPTHPGD
SCHEMBL8037833 0.80 SMO (0.39) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8040180 0.80 S1PR1 (0.58) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8038215 0.79 S1PR1 (0.40) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8041698 0.79 CYP1A2 (0.41) S1PR1KDM4ELMNACYP3A4MAPT
SCHEMBL8041701 0.79 APP (0.38) S1PR1LMNAMAPTGAAAPP
SCHEMBL8033842 0.77 RAB9A (0.42) S1PR1CYP3A4MAPTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed