SCHEMBL8037447

SCHEMBL8037447

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NC(C)(C)C)cc1O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 7/20 0.41
KDM4E B2RXH2 4/20 0.41
GAA P10253 1/20 0.41
APP P05067 1/20 0.39
PYGL P06737 3/20 0.38
ADRB2 P07550 1/20 0.37
GPR183 P32249 1/20 0.37
APLNR P35414 1/20 0.37
S1PR5 Q9H228 1/20 0.37
PTPN7 P35236 1/20 0.37
DUSP3 P51452 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 2/20 0.36
TMPRSS4 Q9NRS4 1/20 0.36
NTRK1 P04629 1/20 0.35
YES1 P07947 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037438 0.84 S1PR1 (0.45) S1PR1KDM4EGAAAPPADRB2
SCHEMBL8039185 0.82 PYGL (0.49) KDM4EGAAPYGLMAPTMAPK1
SCHEMBL8040252 0.81 ALDH1A1 (0.41) S1PR1KDM4EGAAMAPT
SCHEMBL8037415 0.81 S1PR1 (0.41) S1PR1GAAAPPADRB2GPR183
SCHEMBL8041411 0.81 S1PR1 (0.43) S1PR1KDM4EAPPMAPT
SCHEMBL8025554 0.81 MTNR1A (0.42) S1PR1KDM4EAPPAURKB
SCHEMBL8040180 0.81 S1PR1 (0.58) S1PR1KDM4EPYGLADRB2GPR183
SCHEMBL8028301 0.81 APP (0.39) S1PR1KDM4EGAAAPPADRB2
SCHEMBL8037435 0.80 PDE10A (0.41) S1PR1APP
SCHEMBL8037394 0.80 POLB (0.46) S1PR1KDM4EGAAAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed