Lirexapride

Lirexapride

SCHEMBL384567

CC1CCN(C[C@H]2CCCC[C@H]2NC(=O)c2cc(Cl)c(N)cc2OCC2CC2)CC1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.50
ACHE P22303 3/20 0.50
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9460481 0.89 HTR4 (0.61) HTR4ACHEDRD2DRD4DRD3
SCHEMBL9460469 0.89 HTR4 (0.61) HTR4ACHEDRD2DRD4DRD3
SCHEMBL9460473 0.89 HTR4 (0.61) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460956 0.88 HTR4 (0.60) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460955 0.88 HTR4 (0.60) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460954 0.88 HTR4 (0.60) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460967 0.88 MAPK1 (0.59) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460964 0.88 MAPK1 (0.59) HTR4ACHEDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9460962 0.88 MAPK1 (0.59) HTR4ACHEDRD2DRD4DRD3
SCHEMBL8052736 0.83 HTR4 (0.52) HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 598 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2956450-B1 HYDROXYINDALPINE DERIVATIVES AND THEIR MEDICAL USE UNIV MUENCHEN TECH (DE) 2018-07-25 EP claimed
US-20150376164-A1 HYDROXYINDALPINE DERIVATIVES AND THEIR MEDICAL USE TECHNISCHE UNIVERSITAT MUNCHEN (DE) 2015-12-31 US claimed
EP-2956450-A1 HYDROXYINDALPINE DERIVATIVES AND THEIR MEDICAL USE Technische Universität München (DE) 2015-12-23 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
WO-2014125084-A1 HYDROXYINDALPINE DERIVATIVES AND THEIR MEDICAL USE Technische Universität München (DE) 2014-08-21 WO claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
WO-2009018169-A1 SUBSTITUTED CYCLOHEXANOLS AUSPEX PHARMACEUTICALS, INC. (US) 2009-02-05 WO claimed
US-20090028873-A1 SUBSTITUTED CYCLOHEXANOLS AUSPEX PHARMACEUTICALS, INC. (US) 2009-01-29 US claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20060241134-A1 Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility ALTANA PHARMA GA (DE) 2006-10-26 US claimed
EP-1644043-A1 PHARMACEUTICAL COMBINATIONS OF A PROTON PUMP INHIBITOR AND A COMPOUND WHICH MODIFIES GASTROINTESTINAL MOTILITY ALTANA Pharma AG (DE) 2006-04-12 EP claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
WO-2005074931-A1 PHARMACEUTICAL COMBINATIONS COMPRISING (S) -PANTOPRAZOLE ALTANA PHARMA AG (DE) 2005-08-18 WO claimed
WO-2004105795-A1 PHARMACEUTICAL COMBINATIONS OF A PROTON PUMP INHIBITOR AND A COMPOUND WHICH MODIFIES GASTROINTESTINAL MOTILITY ALTANA PHARMA AG (DE) 2004-12-09 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150376164-A1 HYDROXYINDALPINE DERIVATIVES AND THEIR MEDICAL USE HTR5A, HTR4, HTR6 HTR4 2/4885ACHE 196/4885DRD2 32/4885
US-20090028873-A1 SUBSTITUTED CYCLOHEXANOLS OPRM1, OPRD1, OPRK1 HTR4 171/4885ACHE 395/4885DRD2 160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.