SCHEMBL8040415

SCHEMBL8040415

O=C1c2ccccc2C(=O)N1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.64
HTR1A P08908 2/20 0.62
HTR2A P28223 2/20 0.62
DRD3 P35462 2/20 0.62
HTR6 P50406 2/20 0.62
HTR7 P34969 1/20 0.62
KCNH2 Q12809 1/20 0.62
ACHE P22303 1/20 0.61
HTR2C P28335 1/20 0.60
ADRA1A P35348 1/20 0.60
HRH1 P35367 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9075983 0.94 ACHE (0.62) DRD2HTR1AHTR2ADRD3HTR6
SCHEMBL793140 0.87 DRD2 (0.70) DRD2HTR1AHTR2AACHEHTR2C
SCHEMBL791048 0.87 DRD2 (0.70) DRD2HTR1AHTR2AHTR6HTR7
Hydrochloric Acid SCHEMBL9596033 0.86 DRD2 (0.69) DRD2HTR1AHTR2AHTR6HTR7
SCHEMBL1544931 0.85 ACHE (0.71) DRD2HTR1AHTR2AACHEHTR2C
Hydrochloric Acid SCHEMBL1545126 0.84 ACHE (0.70) DRD2HTR1AHTR2AACHEHTR2C
SCHEMBL1545461 0.83 HTR1A (0.76) DRD2HTR1AHTR2ADRD3HTR6
SCHEMBL5995122 0.81 HTR1A (0.67) DRD2HTR1AHTR2A
SCHEMBL7355139 0.81 ACHE (0.68) DRD2HTR1AHTR2ADRD3HTR6
SCHEMBL1545289 0.81 ACHE (0.65) DRD2HTR1AHTR2AACHEHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043240-A USEFUL AS ANTIPSYCHOTIC AND ANALGESIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 2000-03-28 US disclosed