SCHEMBL8040824

SCHEMBL8040824

O=C(O)C(=O)/C=C(\O)c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.67
CA2 P00918 4/20 0.67
CA12 O43570 2/20 0.67
CA9 Q16790 2/20 0.67
CYP1A2 P05177 1/20 0.66
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
BCL2L1 Q07817 1/20 0.47
BAD Q92934 1/20 0.47
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 1/20 0.42
NFE2L2 Q16236 1/20 0.42
PTPN1 P18031 1/20 0.41
TNFRSF1A P19438 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040828 1.00 CA1 (0.67) CA1CA2CA12CA9CYP1A2
SCHEMBL13864066 0.81 NFE2L2 (0.65) CA1CA2CYP1A2CES2CES1
SCHEMBL6662254 0.80 CA12 (1.00) CA1CA2CA12CA9CYP1A2
SCHEMBL8364933 0.80 MAPT (0.73) CA1CA2CA12CA9CYP1A2
SCHEMBL8364930 0.80 MAPT (0.73) CA1CA2CA12CA9CYP1A2
SCHEMBL7378257 0.79 CA1 (0.67) CA1CA2CA12CA9CYP1A2
SCHEMBL12168638 0.79 MAPT (0.48) CA1CA2CA12CA9CYP1A2
SCHEMBL7378259 0.79 CA1 (0.67) CA1CA2CA12CA9CYP1A2
SCHEMBL8029219 0.79 ALDH1A1 (0.68) CA1CA2CA12CA9CYP1A2
SCHEMBL8029217 0.79 ALDH1A1 (0.68) CA1CA2CA12CA9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0868420-B1 3-PYRAZOLECARBOXAMIDE DERIVATIVES HAVING CANNABINOID RECEPTOR AFFINITY SANOFI SYNTHELABO (FR) 2000-03-29 EP disclosed
EP-0885889-A2 Process for the preparation of pyrazole-3-carboxylic acids SANOFI (FR) 1998-12-23 EP disclosed
EP-0868420-A1 3-PYRAZOLECARBOXAMIDE DERIVATIVES HAVING CANNABINOID RECEPTOR AFFINITY SANOFI (FR) 1998-10-07 EP disclosed
WO-1997021682-A1 3-PYRAZOLECARBOXAMIDE DERIVATIVES HAVING CANNABINOID RECEPTOR AFFINITY SANOFI (FR) 1997-06-19 WO disclosed