Phenoperidine

Phenoperidine

SCHEMBL80415

CCOC(=O)C1(c2ccccc2)CCN(CCC(O)c2ccccc2)CC1

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 3/20 0.83
OPRM1 P35372 9/20 0.70
OPRD1 P41143 7/20 0.70
OPRK1 P41145 6/20 0.70
SLC22A1 O15245 1/20 0.66
SLC6A4 P31645 1/20 0.66
ADRA1A P35348 1/20 0.66
KCNH2 Q12809 1/20 0.66
MEN1 O00255 1/20 0.56
LMNA P02545 1/20 0.56
KMT2A Q03164 1/20 0.56
TDP1 Q9NUW8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenoperidine SCHEMBL394330 0.99 KCNA3 (0.81) KCNA3OPRM1OPRD1OPRK1SLC22A1
Phenoperidine SCHEMBL1652634 0.98 KCNA3 (0.80) KCNA3OPRM1OPRD1OPRK1SLC22A1
Phenoperidine SCHEMBL28832646 0.89 KCNA3 (0.67) KCNA3OPRM1OPRD1OPRK1SLC22A1
Oxpheneridine SCHEMBL2110574 0.88 OPRM1 (0.73) KCNA3OPRM1OPRD1OPRK1SLC22A1
SCHEMBL8188731 0.84 KCNA3 (0.58) KCNA3SLC6A4KMT2A
SCHEMBL11712840 0.84 OPRM1 (0.82) KCNA3OPRM1OPRD1OPRK1SLC22A1
SCHEMBL11601769 0.83 OPRM1 (0.80) KCNA3OPRM1OPRD1OPRK1SLC22A1
SCHEMBL11712071 0.83 OPRM1 (1.00) KCNA3OPRM1OPRD1OPRK1SLC22A1
Phenoperidine SCHEMBL3992197 0.82 OPRM1 (0.61) KCNA3OPRM1OPRD1OPRK1SLC22A1
SCHEMBL8216361 0.82 KCNA3 (0.56) KCNA3SLC6A4ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7535 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-20250319074-A1 TREATMENT AND MANAGEMENT OF AUGMENTATION IN RESTLESS LEGS SYNDROME UNIV EAST CAROLINA (US) 2025-10-16 US claimed
US-12383743-B2 Treatment of addiction and dependency TACA JR ARTURO C (US) 2025-08-12 US claimed
US-20250228771-A1 ALKALINE INTRAORAL PRODUCTS EMPLICURE AB (publ) (SE) 2025-07-17 US claimed
EP-4581017-A1 NEW N-HETEROARYLBENZAMIDES DERIVATIVES AS FLT3 INHIBITORS Biodol Therapeutics (FR) 2025-07-09 EP claimed
EP-4565202-A1 ALKALINE INTRAORAL PRODUCTS EMPLICURE AB (publ) (SE) 2025-06-11 EP claimed
WO-2024254056-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF CATALENT ONTARIO LIMITED (CA) 2024-12-12 WO claimed
US-12133922-B2 Abuse resistant capsule R.P. SCHERER TECHNOLOGIES, LLC (US) 2024-11-05 US claimed
US-20240288374-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation 2024-08-29 US claimed
WO-2024172892-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation (US) 2024-08-22 WO claimed
CN-1130352-A Method for relieving pain by orally administering 24-hour sustained-release opioid dosage form capable of rapidly increasing initial blood concentration of patient EURO CELTIQUE SA (LU) 1996-09-04 CN claimed
WO-1996014058-A1 MELT-EXTRUDED ORALLY ADMINISTRABLE OPIOID FORMULATIONS EURO-CELTIQUE, S.A. (LU) 1996-05-17 WO claimed
WO-1995014460-A1 OPIOID FORMULATIONS FOR TREATING PAIN EURO-CELTIQUE S.A. (LU) 1995-06-01 WO claimed
EP-0647448-A1 Orally administrable opioid formulations having extended duration of effect Euroceltique S.A. (LU) 1995-04-12 EP claimed
EP-0341745-B1 Crosslinked carboxy polysaccharides FIDIA SPA (IT) 1994-12-14 EP claimed
EP-0608893-A1 Inhibiting the development of tolerance to and/or dependence on an additive substance VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-08-03 EP claimed
EP-0376999-A1 METHOD OF REVERSING THE SIDE EFFECTS OF EPIDURAL ANALGESICS BAKER CUMMINS PHARMACEUTICALS, INC. (US) 1990-07-11 EP claimed
WO-1989010125-A1 METHOD OF REVERSING THE SIDE EFFECTS OF EPIDURAL ANALGESICS BAKER CUMMINS PHARMACEUTICALS, INC (US) 1989-11-02 WO claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed
US-4053604-A 3-HYDROXY-3-ISOPROPYL-2,3,4,4A,8,9,13B,14-OCTAHYDRO-1H -BENZO(6,7)CYCLOPENTA(1,2,3-DE)PYRIDO(2,1-A)ISOQUINOLIN-3-OL AYERST, MCKENNA & HARRISON LIMITED (CA) 1977-10-11 US claimed