SCHEMBL8042378

SCHEMBL8042378

Cn1nnc(Sc2nc(-c3ccccc3)cs2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.47
HTR2A P28223 1/20 0.47
HTR7 P34969 1/20 0.47
RAB9A P51151 7/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 3/20 0.44
ALDH1A1 P00352 5/20 0.43
HSD17B10 Q99714 3/20 0.43
NPC1 O15118 4/20 0.42
TDP1 Q9NUW8 2/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
AR P10275 3/20 0.41
TP53 P04637 2/20 0.41
ALOX15 P16050 2/20 0.41
HPGD P15428 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
GFER P55789 1/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033890 0.86 RAB9A (0.46) RAB9AHTTMAPTALDH1A1HSD17B10
SCHEMBL8051868 0.84 HTR1A (0.52) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8034092 0.84 HTR1A (0.49) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8046620 0.82 RAB9A (0.44) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8043826 0.82 HTR1A (0.44) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8043683 0.82 HTR1A (0.47) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8048789 0.80 HTR1A (0.45) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8032624 0.80 RAB9A (0.49) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8047618 0.78 RAB9A (0.46) HTR1AHTR2AHTR7RAB9AHTT
SCHEMBL8048790 0.77 RAB9A (0.44) HTR1AHTR2AHTR7RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed