SCHEMBL8042407

SCHEMBL8042407

CS(=O)(=O)c1cnc(Sc2nnnn2-c2ccc(S(N)(=O)=O)cc2)s1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.43
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712725 0.92 PTGS2 (0.39) PTGS2ALDH1A1HSD17B10LMNATP53
SCHEMBL8050190 0.87 ALDH1A1 (0.40) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8048309 0.86 ALDH1A1 (0.52) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8033930 0.86 ALDH1A1 (0.39) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8046366 0.85 PTGS2 (0.50) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8042987 0.85 PTGS2 (0.50) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8042077 0.85 ALDH1A1 (0.39) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8032741 0.84 PTGS2 (0.48) PTGS2ALDH1A1HSD17B10HPGDLMNA
SCHEMBL8041899 0.84 RECQL (0.49) ALDH1A1HSD17B10HPGDLMNATP53
SCHEMBL8049857 0.83 EP300 (0.44) PTGS2ALDH1A1HSD17B10HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed