SCHEMBL8032741

SCHEMBL8032741

NS(=O)(=O)c1ccc(-n2nnnc2Sc2ncc(Cl)s2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.48
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
HSD17B10 Q99714 4/20 0.39
ALDH1A1 P00352 4/20 0.39
TP53 P04637 3/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 2/20 0.39
MAPK1 P28482 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39
PTGS1 P23219 4/20 0.38
JAK2 O60674 1/20 0.38
TLR9 Q9NR96 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042407 0.84 PTGS2 (0.43) PTGS2CA12CA1CA2CA9
SCHEMBL8050630 0.84 MAPK8 (0.46) PTGS2ALDH1A1MAPTMAPK1KMT2A
SCHEMBL8048031 0.84 PTGS2 (0.45) PTGS2CA12CA1CA2CA9
SCHEMBL8045773 0.82 EP300 (0.45) CA1CA2CA9HSD17B10ALDH1A1
SCHEMBL8042845 0.82 ALDH1A1 (0.42) HSD17B10ALDH1A1TP53HPGDMAPT
SCHEMBL8043646 0.82 ALDH1A1 (0.54) HSD17B10ALDH1A1TP53HPGDMAPT
SCHEMBL8046903 0.81 HPGD (0.50) HSD17B10ALDH1A1TP53HPGDMAPT
SCHEMBL8044972 0.80 ALDH1A1 (0.43) HSD17B10ALDH1A1TP53HPGDMAPT
SCHEMBL8042672 0.79 ALDH1A1 (0.42) PTGS2HSD17B10ALDH1A1TP53HPGD
SCHEMBL8044841 0.79 KDM4E (0.49) HSD17B10ALDH1A1TP53HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed