SCHEMBL8042672

SCHEMBL8042672

CN(C)c1ccc(-n2nnnc2Sc2ncc(Cl)s2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.42
MAPT P10636 7/20 0.42
HSD17B10 Q99714 5/20 0.42
TP53 P04637 5/20 0.42
KMT2A Q03164 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MAPK1 P28482 4/20 0.42
KDM4E B2RXH2 4/20 0.42
NPSR1 Q6W5P4 3/20 0.42
TSHR P16473 3/20 0.42
HPGD P15428 2/20 0.42
POLB P06746 2/20 0.42
LMNA P02545 7/20 0.41
HTT P42858 4/20 0.41
PTGS2 P35354 2/20 0.40
JAK2 O60674 1/20 0.39
TLR9 Q9NR96 1/20 0.39
MEN1 O00255 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044972 0.84 ALDH1A1 (0.43) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8042845 0.84 ALDH1A1 (0.42) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8043646 0.84 ALDH1A1 (0.54) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8044841 0.83 KDM4E (0.49) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8042987 0.82 PTGS2 (0.50) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8047631 0.82 MAPT (0.41) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8050651 0.81 MAPT (0.44) ALDH1A1MAPTKMT2ASMN1; SMN2MAPK1
SCHEMBL8046903 0.80 HPGD (0.50) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8032741 0.79 PTGS2 (0.48) ALDH1A1MAPTHSD17B10TP53KMT2A
SCHEMBL8044847 0.79 SMN1; SMN2 (0.45) ALDH1A1MAPTHSD17B10TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed