SCHEMBL8042975

SCHEMBL8042975

CC(C)(C)OC(=O)NC1CCN(CC(O)COc2ccc(F)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.62
SCN1A P35498 1/20 0.57
SCN5A Q14524 1/20 0.57
SCN9A Q15858 1/20 0.57
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP2D6 P10635 3/20 0.52
ABCB1 P08183 3/20 0.52
HTR2A P28223 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
MAPT P10636 2/20 0.50
USP2 O75604 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SSTR4 P31391 1/20 0.49
RECQL P46063 1/20 0.48
CACNA1G O43497 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24225699 0.90 SCN1A (0.55) SCN1ASCN5ASCN9AMEN1KMT2A
SCHEMBL8054546 0.89 SCN1A (0.52) TSHRSCN1ASCN5ASCN9AMEN1
SCHEMBL29356382 0.87 ATF4 (0.58) TSHRSCN1ASCN5ASCN9AUSP2
SCHEMBL4340211 0.83 SCN5A (0.55) TSHRSCN1ASCN5ASCN9AMEN1
SCHEMBL22373890 0.81 ATF4 (0.54) SCN1ASCN5ASCN9A
SCHEMBL7808692 0.81 TSHR (0.75) TSHRMEN1KMT2ACYP2D6ABCB1
Hydrochloric Acid SCHEMBL8055599 0.80 TSHR (0.73) TSHRMEN1KMT2ACYP2D6ABCB1
SCHEMBL621716 0.80 CTSK (0.46) SCN1ASCN5ASCN9A
SCHEMBL5749820 0.80 HTR2A (0.64) TSHRMEN1KMT2AABCB1HTR2A
SCHEMBL3351581 0.78 SIGMAR1 (0.60) CYP2D6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011032-A Heterocyclic compounds for treating myocardial ischemia PIERRE FABRE MEDICAMENT (FR) 2000-01-04 US disclosed