SCHEMBL8043262

SCHEMBL8043262

Oc1c(Br)cc(Br)cc1-c1nnc(S)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.52
GABRB1 P18505 1/20 0.52
GABRA2 P47869 1/20 0.52
GABRB2 P47870 1/20 0.52
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SNCA P37840 1/20 0.36
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
ERN1 O75460 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PLG P00747 1/20 0.33
PLAU P00749 1/20 0.33
PLAT P00750 1/20 0.33
PRSS1 P07477 1/20 0.33
MEN1 O00255 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050870 0.77 MGAM (0.47) TSHRSNCAKMT2ALMNAMAPT
Bromophene SCHEMBL29429127 0.71 GABRA1 (1.00) GABRA1GABRB1GABRA2GABRB2CYP3A4
Bromophene SCHEMBL31323101 0.71 GABRA1 (1.00) GABRA1GABRB1GABRA2GABRB2CYP3A4
Bromophene SCHEMBL2783711 0.71 GABRA1 (1.00) GABRA1GABRB1GABRA2GABRB2CYP3A4
SCHEMBL8043597 0.70 MGAM (0.40) GABRA1GABRA2GABRB2MAPTMGAM
SCHEMBL12666319 0.67 GABRA1 (0.57) GABRA1GABRB1GABRA2GABRB2CYP3A4
SCHEMBL30471834 0.66 RAB9A (0.60) GABRA1GABRB1GABRA2GABRB2TDP1
SCHEMBL7197008 0.66 RAB9A (0.60) GABRA1GABRB1GABRA2GABRB2TDP1
SCHEMBL18224 0.63 CYP3A4 (1.00) GABRA1GABRB1GABRA2GABRB2CYP3A4
SCHEMBL8047389 0.63 CA1 (0.49) SNCALMNAMGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed