SCHEMBL8043350

SCHEMBL8043350

C=CCN(CC=C)c1c(C)c(C)cc(N)c1N

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 2/20 0.33
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18096367 0.71 CRHR1 (0.47) CRHR1
SCHEMBL11129148 0.68 CYP3A4 (0.38) CRHR1CYP3A4
SCHEMBL6580919 0.67 S100B (0.62) CRHR1CYP3A4TSHR
SCHEMBL11376288 0.64 CRHR1 (0.33) CRHR1
SCHEMBL1050286 0.64 USP2 (0.33) TSHR
SCHEMBL9153229 0.63 S100B (0.72) CRHR1CYP3A4TSHRMAPK1
SCHEMBL14328255 0.63 ESR1 (0.37) CRHR1CYP3A4TSHRMAPK1
SCHEMBL11045130 0.63 CYP3A4 (0.39) CYP3A4TSHR
SCHEMBL2120713 0.63 CYP3A4 (0.48) CYP3A4TSHRMAPK1
SCHEMBL476444 0.63 CYP3A4 (0.48) CYP3A4TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6110911-A ADMINISTERING NEUROPROTECTANT/ANTICONVULSANT TO PATIENT WARNER-LAMBERT COMPANY (US) 2000-08-29 US disclosed
US-5874426-A USEFUL IN THE TREATMENT OF STROKE, CEREBRAL ISCHEMIA, OR CEREBRAL INFARCTION RESULTING FROM THROMBOEMBOLIC OR HEMORRHAGIC STROKE, CEREBRAL VASOSPASMS, HYPOGLYCEMIA, CARDIAC ARREST, STATUS EPILEPTICUS, ANOXIA, SEIZURE DISORDER WARNER-LAMBERT COMPANY (US) 1999-02-23 US disclosed
WO-1996040651-A1 ALKYL AMINE DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1996-12-19 WO disclosed