SCHEMBL8043859

SCHEMBL8043859

CCCC(C)CN(CCN1CCOCC1)c1nc2c(C(C)(C)C)nn(C)c2c(=O)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
PDE9A O76083 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
ALDH1A1 P00352 5/20 0.34
PDE5A O76074 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 2/20 0.34
PDE6C P51160 1/20 0.34
POLB P06746 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
HIF1A Q16665 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
HSD17B10 Q99714 2/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048797 0.90 PDE9A (0.38) KDM4EPDE9APDE1APDE1BPDE1C
SCHEMBL8034133 0.82 KDM4E (0.36) KDM4EPDE9APDE1APDE1BPDE1C
SCHEMBL8044800 0.81 PDE5A (0.44) PDE9APDE1APDE1BPDE1CALDH1A1
SCHEMBL4903611 0.81 KDM4E (0.36) KDM4EPDE9APDE1APDE1BPDE1C
SCHEMBL4906373 0.79 KDM4E (0.43) KDM4EALDH1A1PDE5ANPSR1SMN1; SMN2
SCHEMBL4143162 0.79 GAA (0.42) KDM4EPDE9APDE1APDE1BPDE1C
SCHEMBL8051166 0.79 PDE5A (0.45) PDE9APDE1APDE1BPDE1CALDH1A1
SCHEMBL4904083 0.76 KDM4E (0.48) KDM4EPDE1APDE1BPDE1CALDH1A1
SCHEMBL4123024 0.75 ALDH1A1 (0.36) KDM4EPDE9APDE1APDE1BPDE1C
SCHEMBL8043292 0.75 PDE5A (0.45) PDE9APDE1APDE1BPDE1CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed