SCHEMBL8048797

SCHEMBL8048797

CC(C)CN(CCN1CCOCC1)c1nc2c(C(C)(C)C)nn(C)c2c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE1C Q14123 1/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 9/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
POLB P06746 3/20 0.34
PDE5A O76074 2/20 0.33
PDE6C P51160 1/20 0.33
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32
HIF1A Q16665 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
GAA P10253 1/20 0.32
USP2 O75604 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043859 0.90 KDM4E (0.36) PDE9APDE1APDE1BPDE1CKDM4E
SCHEMBL8034133 0.86 KDM4E (0.36) PDE9APDE1APDE1BPDE1CKDM4E
SCHEMBL8051166 0.84 PDE5A (0.45) PDE9APDE1APDE1BPDE1CALDH1A1
SCHEMBL4143162 0.82 GAA (0.42) PDE9APDE1APDE1BPDE1CKDM4E
SCHEMBL4123024 0.79 ALDH1A1 (0.36) PDE9APDE1APDE1BPDE1CKDM4E
SCHEMBL4131950 0.77 GAA (0.41) PDE9APDE1APDE1BPDE1CKDM4E
SCHEMBL4901385 0.77 KDM4E (0.44) KDM4EALDH1A1SMN1; SMN2MAPTNPSR1
SCHEMBL8044800 0.77 PDE5A (0.44) PDE9APDE1APDE1BPDE1CALDH1A1
SCHEMBL4134627 0.76 MAPT (0.34) KDM4EALDH1A1MAPTNPSR1POLB
SCHEMBL8042659 0.76 KDM4E (0.37) KDM4EALDH1A1SMN1; SMN2MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed