SCHEMBL8044945

SCHEMBL8044945

CCNC(=O)ONC(=O)CCCCCC(C#N)(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 6/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
KCNH2 Q12809 1/20 0.40
OPRM1 P35372 4/20 0.39
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
CYP2D6 P10635 1/20 0.39
HDAC6 Q9UBN7 2/20 0.37
CCR1 P32246 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
EPHX2 P34913 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045183 0.86 OPRM1 (0.43) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8044965 0.86 OPRM1 (0.43) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8045058 0.85 CYP3A4 (0.52) KCNA3CYP3A4CYP2C9KCNH2HDAC6
SCHEMBL8049747 0.83 CYP3A4 (0.43) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8044655 0.83 CYP3A4 (0.43) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8045765 0.81 CCR1 (0.40) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8035678 0.79 CYP3A4 (0.40) CYP3A4CYP2C9KCNH2CYP2D6HDAC6
SCHEMBL8052908 0.78 KMT2A (0.40) KCNA3CYP3A4CYP2C9KCNH2OPRM1
SCHEMBL8035137 0.78 HDAC1 (0.51) CYP3A4KCNH2HDAC6HDAC3HDAC4
SCHEMBL8035139 0.78 HDAC1 (0.51) CYP3A4KCNH2HDAC6HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed