SCHEMBL8045183

SCHEMBL8045183

CCC(=O)ONC(=O)CCCCCC(C#N)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
DRD3 P35462 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
KCNH2 Q12809 1/20 0.42
KCNA3 P22001 6/20 0.41
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CCR1 P32246 2/20 0.38
CCR3 P51677 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044965 1.00 OPRM1 (0.43) OPRM1DRD2DRD4DRD3CYP2D6
SCHEMBL8045765 0.94 CCR1 (0.40) OPRM1DRD2DRD4DRD3CYP2D6
SCHEMBL8050105 0.90 HDAC3 (0.38) OPRM1KCNA3RAB9AHDAC6
SCHEMBL8052916 0.89 HDAC6 (0.41) CYP2D6CYP3A4CYP2C9KCNH2CCR1
SCHEMBL8044769 0.89 GAA (0.39) CCR1HDAC6
SCHEMBL8035359 0.88 ALDH1A1 (0.41) CCR1HDAC6
SCHEMBL8044945 0.86 KCNA3 (0.41) OPRM1DRD2DRD4DRD3CYP2D6
SCHEMBL8049785 0.86 HDAC1 (0.37) OPRM1DRD2DRD4DRD3CYP2D6
SCHEMBL8049690 0.86 HDAC6 (0.36) CYP3A4CYP2C9KCNH2KCNA3RAB9A
SCHEMBL8044655 0.85 CYP3A4 (0.43) OPRM1DRD2DRD4DRD3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP claimed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US claimed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP claimed
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed