SCHEMBL8044956

SCHEMBL8044956

CCOC(=O)C(CCCCC(C#N)c1ccccc1)c1nccs1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CTSA P10619 14/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PKM P14618 1/20 0.40
MMP8 P22894 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050089 0.82 SMN1; SMN2 (0.58) MEN1GAAKMT2ASMN1; SMN2CYP1A2
SCHEMBL4330530 0.74 CTSA (0.43) CTSACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9705564 0.72 CYP3A4 (0.49) MEN1GAAKMT2ASMN1; SMN2CYP1A2
SCHEMBL4327564 0.71 CTSA (0.43) CTSACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4334693 0.71 CTSA (0.43) CTSACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4325302 0.70 FPR2 (0.38) MEN1KMT2ACTSACYP1A2CYP3A4
SCHEMBL4329554 0.69 CTSA (0.43) CTSAPKM
SCHEMBL4322245 0.69 SLC6A9 (0.45) CTSACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4332670 0.69 SLC6A9 (0.45) CTSACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4331310 0.69 CTSA (0.43) CTSAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed