SCHEMBL8045101

SCHEMBL8045101

COC(=O)c1cc2c(cc1C)CC(C)S2(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.39
KDM4E B2RXH2 6/20 0.39
HPGD P15428 5/20 0.39
MAPT P10636 3/20 0.39
GAA P10253 2/20 0.39
HSD17B10 Q99714 2/20 0.39
GLA P06280 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
ATM Q13315 1/20 0.39
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057108 0.83 MEN1 (0.34) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8060713 0.82 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8063047 0.81 CFTR (0.39) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8060654 0.80 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8057307 0.79 CHRNB2 (0.44) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8062974 0.78 CA2 (0.37) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8056948 0.77 ALDH1A1 (0.33) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8058228 0.77 ALDH1A1 (0.37) ALDH1A1KDM4EHPGDMAPTGAA
SCHEMBL8062871 0.77
SCHEMBL8063021 0.74 LMNA (0.40) ALDH1A1KDM4EHPGDMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed