SCHEMBL8045260

SCHEMBL8045260

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CC(C)(C)O2

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.33
KDM4E B2RXH2 9/20 0.33
HSD17B10 Q99714 4/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 5/20 0.33
TSHR P16473 4/20 0.33
RAB9A P51151 3/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 2/20 0.33
LMNA P02545 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060677 0.85 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10MAPTKMT2A
SCHEMBL8056991 0.81 ALDH1A1 (0.33) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8057324 0.80
SCHEMBL8060815 0.79 KDM4E (0.38) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8062746 0.78 RXRA (0.36) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8056280 0.77 KDM4E (0.43) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8062776 0.77 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8045354 0.76 ALOX5 (0.43) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8057016 0.76 ALDH1A1 (0.35) ALDH1A1KDM4EHSD17B10MAPTHTT
SCHEMBL8062982 0.76 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed