SCHEMBL8045568

SCHEMBL8045568

c1ccc(CNCC2CCc3ccc4c(c3O2)CCC4)cc1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.68
NFKB2 Q00653 1/20 0.68
RELA Q04206 1/20 0.68
DRD2 P14416 15/20 0.65
DRD4 P21917 15/20 0.65
DRD3 P35462 15/20 0.65
DRD1 P21728 2/20 0.58
DRD5 P21918 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312005 0.79 DRD2 (1.00) NFKB1NFKB2RELADRD2DRD4
SCHEMBL7203555 0.77 NFKB1 (0.44) NFKB1NFKB2RELADRD2DRD4
SCHEMBL8864198 0.77 DRD2 (0.72) NFKB1NFKB2RELADRD2DRD4
SCHEMBL5640879 0.77 DRD2 (0.72) NFKB1NFKB2RELADRD2DRD4
SCHEMBL8864160 0.77 DRD2 (0.72) NFKB1NFKB2RELADRD2DRD4
Bromide SCHEMBL6281511 0.76 DRD2 (0.70) NFKB1NFKB2RELADRD2DRD4
SCHEMBL7116091 0.74 NFKB1 (0.57) NFKB1NFKB2RELADRD2DRD4
SCHEMBL7116097 0.74 NFKB1 (0.57) NFKB1NFKB2RELADRD2DRD4
SCHEMBL8844842 0.73 DRD2 (1.00) DRD2DRD4DRD3DRD1DRD5
SCHEMBL6049929 0.73 HTR1A (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100268-A MIGRAINES JANSSEN PHARMACEUTICA, N.V. (BE) 2000-08-08 US disclosed
EP-0714396-A1 VASOCONTRICTIVE DIHYDROBENZOPYRAN DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1996-06-05 EP disclosed
WO-1995005383-A1 VASOCONTRICTIVE DIHYDROBENZOPYRAN DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1995-02-23 WO disclosed