SCHEMBL8046052

SCHEMBL8046052

N#CCc1ccccc1-c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.41
PTGS1 P23219 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.40
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
DPP4 P27487 1/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
SQOR Q9Y6N5 3/20 0.38
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
NR4A2 P43354 1/20 0.37
HTR7 P34969 1/20 0.37
ACHE P22303 1/20 0.36
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27486706 0.85 PTGS2 (0.38) PTGS2PTGS1ALDH1A1HPGDPTGDR2
SCHEMBL1443804 0.84 GRIA1 (0.39) PTGS2PTGS1ALDH1A1HPGDPTGDR2
SCHEMBL1343377 0.84 DPP4 (0.56) ALDH1A1HPGDDPP4HTR7
SCHEMBL29019013 0.82 TNF (0.47) ALDH1A1HPGDFFAR1FFAR4DPP4
SCHEMBL29842617 0.82 TNF (0.47) ALDH1A1HPGDFFAR1FFAR4DPP4
SCHEMBL4666102 0.81 ESR2 (0.56) ALDH1A1HPGDDPP4ADORA1
SCHEMBL7013171 0.81 HTR7 (0.42) ALDH1A1HPGDFFAR1FFAR4DPP4
SCHEMBL554701 0.81 CYP2C19 (0.45) PTGS2PTGS1ALDH1A1HPGDPTGDR2
SCHEMBL1041243 0.78 PDK2 (0.49) PTGS2PTGS1PTGDR2FFAR1FFAR4
SCHEMBL28812241 0.77 KCNA5 (0.51) PTGS1ALDH1A1HPGDDPP4SQOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed