SCHEMBL8046739

SCHEMBL8046739

O=C(CCCCc1ccnc2ccccc12)C1C2CCC(C2)N1S(=O)(=O)CC1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.35
IDO1 P14902 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
PREP P48147 1/20 0.34
CHRM1 P11229 2/20 0.33
HDAC6 Q9UBN7 1/20 0.32
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
P2RX7 Q99572 1/20 0.31
FAP Q12884 1/20 0.31
NPY1R P25929 1/20 0.31
NPY5R Q15761 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048468 0.84 HPGD (0.41) SMYD3PREP
SCHEMBL8046810 0.72 SMYD3 (0.35) SMYD3PREP
SCHEMBL8043206 0.72 GRIN2B (0.39) SMYD3PREP
SCHEMBL6706106 0.72 ALDH1A1 (0.42) SMYD3
SCHEMBL8043737 0.69 SMYD3 (0.42) SMYD3
SCHEMBL8043736 0.69 SMYD3 (0.42) SMYD3
SCHEMBL5210378 0.65 CYP1A2 (0.51) HDAC6
SCHEMBL7829170 0.64 MAPT (0.51)
SCHEMBL7832661 0.64 MAPT (0.51)
SCHEMBL8044025 0.64 SMYD3 (0.38) SMYD3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121280-A Azabicyclic rotomase inhibitors PFIZER INC. (US) 2000-09-19 US disclosed
EP-0947506-A1 2-Aza-bicyclo[2.2.1]heptane derivatives and their use as rotamase inhibitors Pfizer Products Inc. (US) 1999-10-06 EP disclosed