SCHEMBL6706106

SCHEMBL6706106

COc1cc(CCCCC(=O)C2C3CCC(C3)N2S(=O)(=O)CC2CCCCC2)cc(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
FKBP1A P62942 9/20 0.41
SIGMAR1 Q99720 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.37
SMYD3 Q9H7B4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8049268 0.84 FKBP1A (0.52) ALDH1A1FKBP1ASIGMAR1KMT2A
SCHEMBL8046810 0.75 SMYD3 (0.35) ALDH1A1TDP1KMT2ASMYD3
SCHEMBL8043206 0.75 GRIN2B (0.39) SMYD3
SCHEMBL8048468 0.75 HPGD (0.41) ALDH1A1KMT2ASMYD3
SCHEMBL8046739 0.72 TACR1 (0.35) SMYD3
SCHEMBL8043737 0.70 SMYD3 (0.42) SMYD3
SCHEMBL8043736 0.70 SMYD3 (0.42) SMYD3
SCHEMBL8044025 0.69 SMYD3 (0.38) ALDH1A1TDP1KMT2ASMYD3
SCHEMBL8044030 0.69 SMYD3 (0.38) ALDH1A1TDP1KMT2ASMYD3
SCHEMBL8048750 0.68 TUBB4A (0.41) ALDH1A1FKBP1ASIGMAR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004010617-A AZA-BICYCLIC ROTOMASE INHIBITOR PFIZER PROD INC 2004-01-15 JP disclosed
US-6121280-A Azabicyclic rotomase inhibitors PFIZER INC. (US) 2000-09-19 US disclosed
EP-0947506-A1 2-Aza-bicyclo[2.2.1]heptane derivatives and their use as rotamase inhibitors Pfizer Products Inc. (US) 1999-10-06 EP disclosed