SCHEMBL8047610

SCHEMBL8047610

O=C(O)Cc1csc(Sc2nnc(-c3cccs3)n2C2CCCCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.46
ALDH1A1 P00352 6/20 0.46
NPSR1 Q6W5P4 3/20 0.46
POLB P06746 2/20 0.46
KDM4E B2RXH2 7/20 0.44
HSD17B10 Q99714 5/20 0.44
HPGD P15428 3/20 0.44
RAB9A P51151 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
TSHR P16473 5/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 2/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050181 0.82 KDM4E (0.46) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8043598 0.81 RECQL (0.55) ALDH1A1NPSR1KDM4EHSD17B10HPGD
SCHEMBL8033896 0.81 NPC1 (0.54) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8043257 0.81 KDM4E (0.43) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8044921 0.78 ALDH1A1 (0.44) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8043612 0.78 HSD17B10 (0.52) ALDH1A1NPSR1KDM4EHSD17B10HPGD
SCHEMBL8043119 0.77 ALDH1A1 (0.48) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8043113 0.77 RAB9A (0.48) GAAALDH1A1NPSR1POLBKDM4E
SCHEMBL8042481 0.77 TSHR (0.52) ALDH1A1NPSR1KDM4EHSD17B10HPGD
SCHEMBL8044125 0.77 KDM4E (0.47) GAAALDH1A1NPSR1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed