SCHEMBL8049026

SCHEMBL8049026

CC(C)(C)n1nnnc1Sc1nc2ccc(S(C)(=O)=O)cc2s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.46
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
ILK Q13418 1/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
ACP1 P24666 1/20 0.39
GAA P10253 1/20 0.39
CA2 P00918 1/20 0.38
POLB P06746 1/20 0.38
CLK1 P49759 2/20 0.38
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033856 0.85 PKM (0.46) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8047478 0.83 PKM (0.44) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8043670 0.83 PKM (0.44) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8045105 0.82 ALDH1A1 (0.40) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8050953 0.82 PDK1 (0.56) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL8033160 0.81 PKM (0.51) PKMALDH1A1SMN1; SMN2KMT2ALMNA
SCHEMBL8042747 0.81 PKM (0.42) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8052304 0.81 ALDH1A1 (0.49) PKMALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8042755 0.80 HCAR3 (0.44) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL8043976 0.79 KDM4E (0.43) PKMALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed