SCHEMBL8049690

SCHEMBL8049690

CCC(=O)ONC(=O)CCCCCC(C#N)(c1ccccc1)c1nccs1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.36
ALOX5 P09917 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CES1 P23141 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.34
HDAC1 Q13547 3/20 0.34
USP2 O75604 2/20 0.33
LMNA P02545 2/20 0.33
MAPK1 P28482 1/20 0.33
NPC1 O15118 1/20 0.33
ADRB2 P07550 1/20 0.33
RAB9A P51151 1/20 0.33
TSHR P16473 1/20 0.33
HDAC3 O15379 1/20 0.33
KCNA3 P22001 1/20 0.33
PLA2G4A P47712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045631 0.88 HDAC6 (0.39) HDAC6ALOX5MEN1KMT2AALDH1A1
SCHEMBL8044965 0.86 OPRM1 (0.43) HDAC6CYP3A4CYP2C9KCNH2RAB9A
SCHEMBL8045183 0.86 OPRM1 (0.43) HDAC6CYP3A4CYP2C9KCNH2RAB9A
SCHEMBL8049980 0.85 HDAC6 (0.50) HDAC6ALOX5CYP3A4KCNH2HDAC1
SCHEMBL8052916 0.84 HDAC6 (0.41) HDAC6CYP3A4CYP2C9KCNH2TSHR
SCHEMBL8035219 0.84 ALOX5 (0.39) ALOX5ALDH1A1CES1KCNA3PLA2G4A
SCHEMBL8045765 0.81 CCR1 (0.40) HDAC6CYP3A4CYP2C9KCNH2HDAC1
SCHEMBL8049785 0.78 HDAC1 (0.37) HDAC6ALDH1A1CYP3A4CYP2C9KCNH2
SCHEMBL8050105 0.77 HDAC3 (0.38) HDAC6KMT2AALDH1A1HDAC1LMNA
SCHEMBL8044769 0.76 GAA (0.39) HDAC6HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed