SCHEMBL8051208

SCHEMBL8051208

Cc1nc2c(OCC3C=CC=CC3)cccn2c(=O)c1CCCl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
ADRA1A P35348 3/20 0.41
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GUCY1B2 O75343 3/20 0.36
GUCY1A2 P33402 3/20 0.36
GUCY1A1 Q02108 3/20 0.36
GUCY1B1 Q02153 3/20 0.36
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964742 0.78 CYP1A2 (0.44) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL8321782 0.77 CYP1A2 (0.42) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL8322317 0.76 ADRA2A (0.44) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL795384 0.75 ATP4A (0.62) HTR1ADRD2HTR2ACYP1A2CYP3A4
SCHEMBL5108689 0.71 KDM4E (0.51) ADRA2AADRA2BADRA2CADRA1A
SCHEMBL28430176 0.70 ENPP2 (0.43) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL900644 0.69 ADRA2A (0.53) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL15095108 0.69 ATP4A (0.62) HTR1ADRD2HTR2ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL900773 0.68 ADRA2A (0.52) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL8323388 0.67 ADRA2A (0.45) ADRA2AADRA2BADRA2CADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045489-A2 PROCESS FOR THE SYNTHESIS OF CMHTP, A PALIPERIDONE INTERMEDIATE TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2009-04-09 WO disclosed