SCHEMBL8051292

SCHEMBL8051292

O=C(O)Cc1csc(Sc2nnnn2-c2cccs2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 3/20 0.38
HSD17B10 Q99714 2/20 0.37
GABRA5 P31644 1/20 0.37
GABRB2 P47870 1/20 0.37
ALDH1A1 P00352 7/20 0.37
PKM P14618 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 3/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPK1 P28482 2/20 0.35
USP2 O75604 1/20 0.35
MAPT P10636 3/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051833 0.85 POLB (0.54) POLBHSD17B10ALDH1A1PKMSMN1; SMN2
SCHEMBL8048121 0.83 ALDH1A1 (0.36) POLBHSD17B10GABRA5GABRB2ALDH1A1
SCHEMBL8043765 0.83 L3MBTL1 (0.41) CYP1A2CYP3A4CYP2D6CYP2C19HSD17B10
SCHEMBL8048414 0.83 LMNA (0.36) POLBHSD17B10GABRA5GABRB2ALDH1A1
SCHEMBL8048131 0.81 MAPK1 (0.43) POLBHSD17B10ALDH1A1PKMSMN1; SMN2
SCHEMBL8044691 0.81 HSD17B10 (0.36) POLBHSD17B10GABRA5GABRB2ALDH1A1
SCHEMBL8043692 0.81 HSD17B10 (0.36) POLBHSD17B10GABRA5GABRB2ALDH1A1
SCHEMBL8034317 0.80 HPGD (0.51) POLBHSD17B10ALDH1A1SMN1; SMN2LMNA
SCHEMBL8041793 0.80 POLB (0.43) POLBHSD17B10GABRA5GABRB2ALDH1A1
SCHEMBL8048242 0.80 HSD17B10 (0.37) POLBHSD17B10GABRA5GABRB2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed