SCHEMBL8052157

SCHEMBL8052157

CCCCOC(=O)NCc1ccc(Br)cc1F

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.47
AKR1B1 P15121 3/20 0.46
AKR1A1 P14550 1/20 0.46
FPR3 P25089 5/20 0.43
FPR2 P25090 5/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FAAH O00519 3/20 0.41
MTNR1B P49286 1/20 0.41
MGLL Q99685 1/20 0.41
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8061592 0.87 P2RX7 (0.52) P2RX7AKR1B1AKR1A1FPR3FPR2
SCHEMBL29925001 0.84 EPHX2 (0.46) FAAHMGLL
SCHEMBL2732148 0.82 FAAH (0.40) CYP2C9CYP2C19FAAH
SCHEMBL8061522 0.82 P2RX7 (0.52) P2RX7AKR1B1AKR1A1FPR3FPR2
SCHEMBL6496382 0.81 ALDH1A1 (0.51)
SCHEMBL18552880 0.80 LMNA (0.45) MTNR1BATM
SCHEMBL7407182 0.79 SMN1; SMN2 (0.53) FPR2CYP2C9CYP2C19
SCHEMBL5729078 0.79 EPHX2 (0.44) CYP2C9CYP2C19FAAH
SCHEMBL8062772 0.78 KMT2A (0.49) P2RX7AKR1B1AKR1A1CYP3A4CYP2C19
SCHEMBL29925442 0.78 SMN1; SMN2 (0.43) CYP2C9CYP2C19FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0764634-B1 N-(4-bromo-2-fluorobenzyl)carbamates and process for their preparation CLARIANT GMBH (DE) 2000-06-14 EP claimed
EP-0764634-A2 N-(4-bromo-2-fluorobenzyl)carbamates and process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-26 EP claimed
EP-1720836-B1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS LILLY CO ELI (US) 2014-04-16 EP disclosed
EP-0764634-B1 N-(4-bromo-2-fluorobenzyl)carbamates and process for their preparation CLARIANT GMBH (DE) 2000-06-14 EP disclosed
EP-0764634-A2 N-(4-bromo-2-fluorobenzyl)carbamates and process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-26 EP disclosed