SCHEMBL8052500

SCHEMBL8052500

NCCCCN1CCc2ccc(Br)cc2C1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.49
DRD3 P35462 2/20 0.46
DRD2 P14416 1/20 0.46
HTR7 P34969 3/20 0.45
PRMT5 O14744 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
ABCB1 P08183 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
MAPT P10636 1/20 0.42
HTR1A P08908 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
PNMT P11086 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979148 0.94 CARM1 (0.49) CARM1DRD3DRD2HTR7PRMT5
SCHEMBL7744214 0.84 DRD2 (0.64) CARM1DRD3DRD2PRMT5L3MBTL1
SCHEMBL4229926 0.80 HTR7 (0.64) DRD3DRD2HTR7HDAC3HDAC1
SCHEMBL6975839 0.79 ABCB1 (0.55) ABCB1
SCHEMBL7844061 0.79 DRD2 (0.74) DRD3DRD2HTR7PRMT5HTR1A
SCHEMBL6980960 0.79 DRD3 (0.43) DRD3DRD2HTR7ABCB1HTR1A
Hydrochloric Acid SCHEMBL4224319 0.78 HTR7 (0.62) DRD3DRD2HTR7L3MBTL1HDAC3
SCHEMBL27921604 0.78 HTR7 (0.62) DRD3DRD2HTR7HDAC3HDAC1
SCHEMBL4225899 0.78 HTR7 (0.62) DRD3DRD2HTR7HDAC3HDAC1
Hydrochloric Acid SCHEMBL4222983 0.78 HTR7 (0.62) DRD3DRD2HTR7L3MBTL1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143762-A DRUGS AS DOPAMINE ANTAGONIST PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM, PLC (GB) 2000-11-07 US disclosed
EP-0922035-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 1999-06-16 EP disclosed
WO-1998006699-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR PHARMACEUTICAL USE SMITHKLINE BEECHAM PLC (GB) 1998-02-19 WO disclosed