SCHEMBL8055375

SCHEMBL8055375

CC(C)(C)c1cccc(C(=O)Cl)c1C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
ALDH1A1 P00352 3/20 0.39
ALOX15 P16050 2/20 0.39
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
ALOX5 P09917 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
ATM Q13315 1/20 0.33
ALOX12 P18054 1/20 0.33
RBP4 P02753 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
CTSS P25774 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30706305 1.00 CA2 (0.43) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL9060838 0.88 ALDH1A1 (0.45) CA2ALDH1A1ALOX15TSHR
SCHEMBL29263958 0.84 CA2 (0.46) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL29678146 0.82 ALOX15 (0.47) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL1434698 0.82 CA2 (0.45) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL273494 0.82 ALOX15 (0.47) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL2154401 0.82 ALDH1A1 (0.48) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL28774188 0.81 CA2 (0.43) CA2ALDH1A1ALOX15GABRA1GABRB2
SCHEMBL28819980 0.81 CA2 (0.43) CA2ALDH1A1GABRA1GABRB2TDP1
SCHEMBL27764801 0.81 ALOX15 (0.46) CA2ALDH1A1ALOX15GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104603105-A Carboxamide or sulfonamide substituted nitrogen-containing 5-membered heterocycles as modulators for the orphan nuclear receptor ROR Gamma PHENEX PHARMACEUTICALS AG 2015-05-06 CN disclosed
EP-0999211-A1 NOVEL PURINE DERIVATIVES AND MEDICINAL USE THEREOF JAPAN ENERGY CORPORATION (JP) 2000-05-10 EP disclosed
CN-1016169-B PROCESS FOR PREPARING IMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 1992-04-08 CN disclosed
CN-88101452-A Imdazole derivatives 1988-10-05 CN disclosed