SCHEMBL8057418

SCHEMBL8057418

CC(C(=O)O)c1cccc(P(=O)(O)Cc2ccccc2O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.45
PTGS2 P35354 5/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 3/20 0.45
CXCR1 P25024 2/20 0.45
CXCR2 P25025 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 2/20 0.45
SLC22A6 Q4U2R8 2/20 0.45
HIF1A Q16665 2/20 0.45
RECQL P46063 1/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPK1 P28482 1/20 0.45
PMP22 Q01453 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CXCL8 P10145 1/20 0.45
THPO P40225 1/20 0.45
HTT P42858 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7609537 0.82 PTGS2 (0.38) PTGS1PTGS2MAPTALDH1A1HPGD
Phosphoric Acid SCHEMBL27934163 0.70 AKR1C3 (0.55) PTGS1PTGS2MAPTALDH1A1HPGD
SCHEMBL20640864 0.70 PGK1 (0.62) PTGS1PTGS2MAPTALDH1A1HPGD
SCHEMBL6037830 0.69 PTGS2 (0.47) PTGS1PTGS2MAPTALDH1A1HPGD
Phosphoric Acid SCHEMBL17156463 0.69 PTGS2 (0.64) PTGS1PTGS2MAPTALDH1A1HPGD
SCHEMBL602096 0.69 PTGS2 (0.69) PTGS1PTGS2MAPTALDH1A1HPGD
Ketoprofen SCHEMBL27575091 0.67 PTGS1 (0.88) PTGS1PTGS2MAPTALDH1A1HPGD
SCHEMBL29627562 0.67 AKR1C3 (0.55) PTGS1PTGS2MAPTALDH1A1HPGD
SCHEMBL10910350 0.67 TSHR (0.51) MAPTALDH1A1HPGDHIF1ACYP3A4
SCHEMBL8061568 0.67 AKR1B1 (0.41) ALDH1A1HPGDLMNAHIF1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046180-A NAALADase inhibitors GUILFORD PHARMACEUTICALS INC. (US) 2000-04-04 US disclosed
EP-0936914-A4 1999-08-25 EP disclosed
EP-0936914-A1 HYDROXY-PHOSPHINYL DERIVATIVES USEFUL AS NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1999-08-25 EP disclosed
WO-1997048400-A1 HYDROXY-PHOSPHINYL DERIVATIVES USEFUL AS NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1997-12-24 WO disclosed