SCHEMBL8057747

SCHEMBL8057747

Cc1ccccc1NC(=O)c1ccc(C2(F)CC2c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.49
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
MAPT P10636 1/20 0.45
POLB P06746 2/20 0.45
HPGD P15428 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
TAS1R2 Q8TE23 1/20 0.45
TP53 P04637 2/20 0.45
THRB P10828 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.42
SSTR3 P32745 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 1/20 0.40
ATM Q13315 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057743 0.91 LMNA (0.47) LMNANPC1RAB9AMAPTPOLB
SCHEMBL8038470 0.89 POLB (0.48) LMNANPC1RAB9AMAPTPOLB
SCHEMBL8054861 0.86 SLC16A3 (0.42) LMNANPC1RAB9AMAPTHPGD
SCHEMBL8040665 0.86 POLB (0.56) LMNANPC1RAB9APOLBHPGD
SCHEMBL8038471 0.86 NPC1 (0.46) LMNANPC1RAB9AMAPTPOLB
SCHEMBL8057750 0.80 RAB9A (0.44) LMNANPC1RAB9APOLBHPGD
SCHEMBL8780006 0.78 NAMPT (0.38) HPGDMEN1KMT2A
SCHEMBL8461900 0.78 TSHR (0.46) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL8055091 0.77 TSHR (0.46) LMNAPOLBSMN1; SMN2ALDH1A1MEN1
SCHEMBL8914972 0.76 LMNA (0.69) LMNANPC1RAB9AMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805795-A1 NOVEL AROMATIC AMIDES, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME, AND USE THEREOF AS PESTICIDES Hoechst Schering AgrEvo S.A. (FR) 1997-11-12 EP claimed
WO-1996022965-A1 NOVEL AROMATIC AMIDES, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME, AND USE THEREOF AS PESTICIDES HOECHST SCHERING AGREVO S.A. (FR) 1996-08-01 WO claimed
US-6013837-A E.G.,4-(2-(3,4,5-TRICHLORO PHENYL) 1-FLUOROCYCLOPROPYL)-N-(2-METHYL PHENYL)BENZAMIDE; PARTICULAR USE AGAINST ARTHROPODS, HELMINTHS AND MOLLUSCS; INSECTICIDES; ACARICIDES; NEMATICIDES; PHOTOSTABILITY; NONTOXIC TO MAMMALS HOECHST MARION ROUSSEL (FR) 2000-01-11 US disclosed
EP-0915831-A1 NOVEL METHOD FOR PREPARING AROMATIC AMIDES AND INTERMEDIATES THEREFOR Hoechst Schering AgrEvo S.A. (FR) 1999-05-19 EP disclosed
WO-1998003470-A1 NOVEL METHOD FOR PREPARING AROMATIC AMIDES AND INTERMEDIATES THEREFOR HOECHST SCHERING AGREVO S.A. (FR) 1998-01-29 WO disclosed
EP-0805795-A1 NOVEL AROMATIC AMIDES, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME, AND USE THEREOF AS PESTICIDES Hoechst Schering AgrEvo S.A. (FR) 1997-11-12 EP disclosed
WO-1996022965-A1 NOVEL AROMATIC AMIDES, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME, AND USE THEREOF AS PESTICIDES HOECHST SCHERING AGREVO S.A. (FR) 1996-08-01 WO disclosed