SCHEMBL8057955

SCHEMBL8057955

COC(=O)[C@H](Cc1ccc(C)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.62
CTSL P07711 2/20 0.61
POLB P06746 2/20 0.60
ATM Q13315 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
MMP9 P14780 6/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CA7 P43166 3/20 0.55
CA12 O43570 2/20 0.55
CA9 Q16790 2/20 0.55
CA14 Q9ULX7 2/20 0.55
CA2 P00918 2/20 0.55
CTSS P25774 1/20 0.55
MMP2 P08253 6/20 0.54
ADAMTS4 O75173 1/20 0.54
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
BACE1 P56817 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14534184 0.95 CTSL (0.67) TDP1CTSLPOLBATML3MBTL1
SCHEMBL20335144 0.95 CTSL (0.67) TDP1CTSLPOLBATML3MBTL1
SCHEMBL20335146 0.95 CTSL (0.67) TDP1CTSLPOLBATML3MBTL1
SCHEMBL27568136 0.92 POLB (0.70) CTSLPOLBMMP9MEN1KMT2A
SCHEMBL26606026 0.91 MMP9 (0.69) TDP1CTSLPOLBMMP9MEN1
SCHEMBL26606022 0.91 MMP9 (0.69) TDP1CTSLPOLBMMP9MEN1
SCHEMBL13226933 0.90 POLB (0.60) CTSLPOLBATML3MBTL1MMP9
SCHEMBL7984123 0.90 POLB (0.60) CTSLPOLBL3MBTL1MMP9MEN1
SCHEMBL7981960 0.88 TDP1 (0.60) TDP1CTSLPOLBATML3MBTL1
SCHEMBL8063645 0.88 TDP1 (0.78) TDP1POLBL3MBTL1MMP9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009042092-A1 2-ARYL OR HETEROARYL INDOLE DERIVATIVES MERCK & CO., INC. (US) 2009-04-02 WO disclosed