SCHEMBL8058494

SCHEMBL8058494

O=C(O)C(CCc1cccs1)(c1ccccc1)[PH](=O)O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
HPGD P15428 2/20 0.38
POLB P06746 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 2/20 0.38
LMNA P02545 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
TSHR P16473 1/20 0.36
RIPK1 Q13546 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059273 0.86 CYP2C19 (0.41) CYP2C19HPGDPOLBTDP1SMN1; SMN2
SCHEMBL8059180 0.77 GRM2 (0.45) POLBTAAR1
SCHEMBL7644315 0.72 GRM2 (0.44) TDP1SMN1; SMN2RAB9ANPC1
SCHEMBL8059183 0.72 CYP1A2 (0.47) CYP2C19HPGDPOLBTDP1SMN1; SMN2
SCHEMBL8046600 0.72 GRM2 (0.41) POLBRAB9ATAAR1
SCHEMBL7633968 0.72 KIF11 (0.43) CYP2C19TDP1RAB9ANPC1LMNA
SCHEMBL4341638 0.71 RIPK1 (0.48) CYP2C19HPGDPOLBTDP1SMN1; SMN2
SCHEMBL4473902 0.71 RIPK1 (0.51) CYP2C19HPGDPOLBTDP1SMN1; SMN2
SCHEMBL8059153 0.71 GRM2 (0.40) POLBRAB9ATAAR1
SCHEMBL7639980 0.71 GAA (0.41) CYP2C19RAB9ANPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046180-A NAALADase inhibitors GUILFORD PHARMACEUTICALS INC. (US) 2000-04-04 US disclosed