SCHEMBL8058893

SCHEMBL8058893

N=C(NC(=O)OCc1ccccc1)c1n[nH]cc1C(=O)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
TDP1 Q9NUW8 3/20 0.45
ATM Q13315 1/20 0.43
POLB P06746 2/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KMT2A Q03164 1/20 0.42
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP12 P39900 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
TSHR P16473 2/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK1 P28482 1/20 0.40
ROCK2 O75116 1/20 0.40
LMNA P02545 2/20 0.40
CASP3 P42574 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777040 0.74 CA12 (0.45) ALDH1A1ATMPOLBHTTROCK2
SCHEMBL7437216 0.73 ALDH1A1 (0.59) ALDH1A1TDP1ATMPOLBKMT2A
SCHEMBL2701264 0.73 ALDH1A1 (0.55) ALDH1A1TDP1POLBSLC6A2SLC6A3
SCHEMBL2321117 0.72 LMNA (0.56) ALDH1A1TDP1POLBSLC6A2SLC6A3
SCHEMBL8775653 0.72 LMNA (0.59) ALDH1A1TDP1POLBSLC6A2SLC6A3
SCHEMBL234454 0.72 LMNA (0.62) ALDH1A1TDP1POLBSLC6A2SLC6A3
SCHEMBL8446295 0.71 SMN1; SMN2 (0.46) ALDH1A1ATMPOLBKMT2AL3MBTL1
SCHEMBL10942377 0.71 LMNA (0.59) TDP1POLBSLC6A2SLC6A3KMT2A
SCHEMBL5845871 0.71 NR4A1 (0.51) TDP1POLBSLC6A2SLC6A3KMT2A
SCHEMBL9788724 0.70 ALDH1A1 (0.68) ALDH1A1TDP1POLBSLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012165-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N- 1- 3- (AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE Aventis Pharmaceuticals Inc. (US) 2000-06-28 EP disclosed
US-5739354-A ONE-STEP GUANYLATION OF 9,6-DIAMINO-5-HYDROXY-4,4-DIFLUORONONANE OR SALT; SIMPLIFICATION, HIGH YIELD END PRODUCT HOECHST MARION ROUSSEL, INC. (US) 1998-04-14 US disclosed
WO-1997035874-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N-[1-[3-[(AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE HOECHST MARION ROUSSEL, INC. (US) 1997-10-02 WO disclosed