SCHEMBL8058952

SCHEMBL8058952

C=CCn1cnc2nc(N)nc(Cl)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.40
ALDH1A1 P00352 1/20 0.37
ADORA2A P29274 5/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ADORA1 P30542 4/20 0.36
SLC2A1 P11166 1/20 0.35
DPP4 P27487 1/20 0.35
HIF1A Q16665 1/20 0.33
HSP90AA1 P07900 4/20 0.33
HSP90AB1 P08238 4/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CCNA1 P78396 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29601777 0.84 ADORA2B (0.39) ADORA2BALDH1A1ADORA2APDE4APDE4B
SCHEMBL9391801 0.79 CSNK2A2 (0.44) ADORA2BALDH1A1ADORA2AADORA1DPP4
SCHEMBL29601416 0.76 ADORA2B (0.40) ADORA2BADORA2AADORA1DPP4HSP90AA1
SCHEMBL2054791 0.76 HSP90AB1 (0.52) HSP90AA1HSP90AB1
SCHEMBL6270755 0.75 ADORA2B (0.46) ADORA2BALDH1A1ADORA2APDE4APDE4B
SCHEMBL170889 0.74 TK1 (0.42) ADORA2BALDH1A1ADORA2APDE4APDE4B
SCHEMBL4846999 0.74 ADORA2A (0.42) ADORA2BALDH1A1ADORA2APDE4APDE4B
SCHEMBL6651365 0.73 ADORA2A (0.32) ADORA2AADORA1
SCHEMBL5659484 0.73 ADORA2B (0.38) ADORA2BALDH1A1ADORA2APDE4APDE4B
SCHEMBL7983989 0.72 ADORA2A (0.35) ALDH1A1ADORA2AADORA1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-07-12 EP disclosed
WO-1999002162-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-01-21 WO disclosed