SCHEMBL8059285

SCHEMBL8059285

COc1ccc([CH]C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
CYP2A6 P11509 1/20 0.52
NFE2L2 Q16236 1/20 0.52
KDM4E B2RXH2 4/20 0.50
CYP3A4 P08684 2/20 0.50
LMNA P02545 2/20 0.50
TP53 P04637 1/20 0.50
TSHR P16473 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
TRPA1 O75762 1/20 0.48
RELA Q04206 1/20 0.48
NQO2 P16083 2/20 0.47
PTGS1 P23219 2/20 0.47
CYP1A2 P05177 3/20 0.47
CYP1A1 P04798 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12471745 0.82 CYP1A2 (0.48) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL9412294 0.79 ALDH1A1 (0.54) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL19787372 0.78 NFE2L2 (0.64) ALDH1A1NFE2L2KDM4ECYP3A4LMNA
SCHEMBL10888408 0.77 ALDH1A1 (0.52) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL5151182 0.75 CHRM5 (0.56) NFE2L2CYP3A4RELANQO2CYP1A2
SCHEMBL17468467 0.74 MAPT (0.54) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL11688441 0.73 ALDH1A1 (0.58) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL154967 0.73 ALDH1A1 (0.58) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL852777 0.73 ALDH1A1 (0.58) ALDH1A1CYP2A6NFE2L2KDM4ECYP3A4
SCHEMBL18144097 0.72 CYP1A1 (0.67) ALDH1A1NFE2L2KDM4ECYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9856275-B2 Synthesis and use of fluorinated compounds THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-01-02 US disclosed
WO-2014126990-A1 SYNTHESIS AND USE OF FLUORINATED COMPOUNDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-08-21 WO disclosed
EP-0758013-B1 Liquid crystalline optical film, compensating film for liquid crystal display and liquid crystal display NIPPON OIL CO LTD (JP) 2000-10-11 EP disclosed
US-6034086-A VIRICIDES; AIDS THERAPY UBE INDUSTRIES, LTD. 2000-03-07 US disclosed
US-5855971-A Liquid crystalline optical film, compensating film for liquid crystal display comprising the liquid crystalline optical film, and liquid crystal display having the compensating film NIPPON OIL COMPANY, LIMITED (JP) 1999-01-05 US disclosed
EP-0758013-A1 Liquid crystalline optical film, compensating film for liquid crystal display and liquid crystal display NIPPON OIL COMPANY, LIMITED (JP) 1997-02-12 EP disclosed
US-4486444-A CARBONIC ANHYDRASE INHIBITORS MERCK & CO., INC. (US) 1984-12-04 US disclosed
US-4477466-A Acyloxy derivatives of [phenylsulfonyl(or sulfinyl)]thiophenesulfonamide for the topical treatment of elevated intraocular pressure MERCK & CO., INC. (US) 1984-10-16 US disclosed